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All peptides
DermatologyResearch Phase

Biopeptide CL (Palmitoyl Tripeptide-5)

Topical
Written by Peptide Association Editorial TeamMedically reviewed by Ian Justl Ellis, MD, CPTLast reviewed Editorial policy

Overview

Palmitoyl Tripeptide-5 is a synthetic lipopeptide consisting of a tripeptide sequence conjugated to palmitic acid to enhance dermal penetration. The peptide is designed to stimulate collagen synthesis by mimicking the activity of thrombospondin-1, a matricellular protein involved in extracellular matrix remodeling.

Mechanism of Action

Its therapeutic rationale centers on attenuating photoaging and improving skin elasticity through upregulation of Types I and III collagen in dermal fibroblasts.

Research Summary & Key Findings

In vitro studies have demonstrated increased collagen gene expression and decreased matrix metalloproteinase activity in cultured human fibroblasts. Small-scale human pilot studies reported improvements in skin roughness and fine lines after 12 weeks of topical application, though peer-reviewed controlled trial data remain limited.

Clinical Status

Research Phase

Biopeptide CL (Palmitoyl Tripeptide-5) is in the research phase with limited clinical data in humans. Current evidence is primarily derived from preclinical (animal or in vitro) studies.

Administration Routes

Topical

References

Primary literature

Study-level citations for this compound are being verified against the primary sources before publication. The database queries above return the current indexed literature in the meantime.

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No lawful pathway today

Biopeptide CL (Palmitoyl Tripeptide-5) is not FDA-approved and does not currently have a lawful prescription or compounding pathway in the United States, so there is nothing for us to sell you here and no consultation to book. That can change: eight peptides moved back to a lawful pathway in February 2026.

Tell me if the status changes

One email, only if this compound's regulatory standing actually moves. Not a newsletter, not a sales sequence.

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Disclaimer: This information is provided for educational and research purposes only. It is not intended as medical advice, diagnosis, or treatment. Always consult a qualified healthcare provider before starting any peptide therapy. The Peptide Association does not endorse or recommend any specific treatment protocol. See our editorial policy for how this content is produced and reviewed.